Molecule Details
InChIKeyLWHTZTIHIFBTMB-UHFFFAOYSA-N
Compound Name1-[6-[5-[5-(methylamino)-1,3,4-thiadiazol-2-yl]-1H-indol-3-yl]-2-pyridinyl]pyrrolidin-2-one
Canonical SMILESCNc1nnc(-c2ccc3[nH]cc(-c4cccc(N5CCCC5=O)n4)c3c2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB