Molecule Details
InChIKeyLVQQMUZNNNCVGV-AREMUKBSSA-N
Compound Name2-[6-[benzyl(methyl)sulfamoyl]-1,3-benzodioxol-5-yl]-N-methyl-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]acetamide
Canonical SMILESCN(C(=O)Cc1cc2c(cc1S(=O)(=O)N(C)Cc1ccccc1)OCO2)[C@H](CN1CCCC1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB