Molecule Details
InChIKeyLVHJAVYIDITWAZ-UHFFFAOYSA-N
Canonical SMILESCC1(C)OB(c2cnc(N)c(-c3cc4cc(NC(=O)Nc5cccc(C(F)(F)F)c5)ccc4s3)c2)OC1(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P09619 PDGFRB Homo sapiens Human PF00047 PF13927 PF25305 PF07714 7.9 IC50 ChEMBL;BindingDB
P35968 KDR Homo sapiens Human PF07679 PF00047 PF13895 PF22971 PF07714 PF21339 PF17988 PF22854 7.9 IC50 ChEMBL;BindingDB