Molecule Details
InChIKeyLVCFJRVHJZAYQL-UHFFFAOYSA-N
Compound Name1-[6-[1-(6-Piperazin-1-yl-2-pyridinyl)pyrazolo[4,3-c]pyridin-6-yl]pyrazin-2-yl]azetidin-3-ol
Canonical SMILESOC1CN(c2cncc(-c3cc4c(cn3)cnn4-c3cccc(N4CCNCC4)n3)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.3 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 10.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.5 Ki ChEMBL;BindingDB