Molecule Details
InChIKeyLVBGEVIMGXRIPY-UHFFFAOYSA-N
Compound Name6-(1H-indol-4-yl)-3-(4-piperazin-1-ylphenyl)-2H-pyrazolo[3,4-b]pyridine
Canonical SMILESc1cc(-c2ccc3c(-c4ccc(N5CCNCC5)cc4)n[nH]c3n2)c2cc[nH]c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB