Molecule Details
InChIKeyLUZBJNWFEDHIPR-LBPRGKRZSA-N
Compound Name(S)-2-(9-(3,4-dichlorophenylthio)-1-isopropyl-7,8-dihydro-6H-pyrido[3,4-b]pyrrolizin-8-yl)acetic acid
Canonical SMILESCC(C)c1nccc2c1c(Sc1ccc(Cl)c(Cl)c1)c1n2CC[C@H]1CC(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13258 PTGDR Homo sapiens Human PF00001 9.2 IC50 ChEMBL;BindingDB
Q9Y5Y4 PTGDR2 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB
P43115 PTGER3 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB