Molecule Details
InChIKeyLUXVBQYXNBNAIG-UHFFFAOYSA-N
Compound Name1-[4-[2-(2-Amino-4-pyridinyl)ethoxy]-3-methoxyphenyl]-3-[3-(5-methylimidazol-1-yl)propyl]-1-(1-methylpiperidin-4-yl)urea
Canonical SMILESCOc1cc(N(C(=O)NCCCn2cncc2C)C2CCN(C)CC2)ccc1OCCc1ccnc(N)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16769 QPCT Homo sapiens Human PF04389 8.4 IC50 ChEMBL;BindingDB
Q9NXS2 QPCTL Homo sapiens Human PF04389 7.7 IC50 ChEMBL;BindingDB