Molecule Details
InChIKeyLUVNXTSNCPCXQE-DZOWNJMZSA-N
Canonical SMILESNC(CCN[C@H](NC(=O)[C@H](Cc1ccc(F)c(F)c1)NC(=O)Nc1ccc2c(CN3CCCC3)cn(Cc3c(Cl)cccc3Cl)c2c1)C(=O)NCc1ccccc1)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25116 F2R Homo sapiens Human PF00001 9.4 Kd ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.5 IC50 ChEMBL;BindingDB