Molecule Details
InChIKeyLUQBIRLUHCYXQM-UHFFFAOYSA-N
Compound Name19-Oxo-2-oxa-9,11,15,18-tetrazapentacyclo[18.6.2.13,7.09,13.024,28]nonacosa-1(27),3,5,7(29),10,12,20,22,24(28),25-decaene-4-carbonitrile
Canonical SMILESN#Cc1ccc2cc1Oc1ccc3cccc(c3c1)C(=O)NCCNCc1cncn1C2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.94
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.3 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.3 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 7.1 IC50 ChEMBL