Molecule Details
InChIKeyLTKYUQAQPQMHNJ-UHFFFAOYSA-N
Compound Name4-[4-Chloro-3-[2-(methylamino)quinazolin-7-yl]oxybenzoyl]-1-methyl-2,5-diphenylpyrazol-3-one
Canonical SMILESCNc1ncc2ccc(Oc3cc(C(=O)c4c(-c5ccccc5)n(C)n(-c5ccccc5)c4=O)ccc3Cl)cc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P2K8 EIF2AK4 Homo sapiens Human PF12745 PF00069 PF05773 PF13393 8.0 IC50 ChEMBL;BindingDB
P15056 BRAF Homo sapiens Human PF00130 PF07714 PF02196 7.9 IC50 ChEMBL;BindingDB
Q9NZJ5 EIF2AK3 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB