Molecule Details
InChIKeyLTKLQMAKAFTREX-UHFFFAOYSA-N
Compound NameN-(4-(4-(naphthalen-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)pyridin-2-yl)cyclopropanecarboxamide
Canonical SMILESO=C(Nc1cc(-c2n[nH]c(=O)n2-c2ccc3ccccc3c2)ccn1)C1CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.64
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB