Molecule Details
InChIKeyLTEDERVMQUPCSO-UHFFFAOYSA-N
Compound Name4-Morpholin-4-yl-6-(3-nitroanilino)-1,3,5-triazine-2-carbonitrile
Canonical SMILESN#Cc1nc(Nc2cccc([N+](=O)[O-])c2)nc(N2CCOCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25774 CTSS Homo sapiens Human PF08246 PF00112 7.7 IC50 ChEMBL;BindingDB
P43235 CTSK Homo sapiens Human PF08246 PF00112 7.0 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.7 IC50 ChEMBL;BindingDB