Molecule Details
InChIKeyLTCOTSRHIWKZTK-NSHDSACASA-N
Compound Name(2S)-2-[[4-[(2-amino-6-methyl-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)sulfanyl]-2-fluorobenzoyl]amino]pentanedioic acid
Canonical SMILESCc1[nH]c2nc(N)[nH]c(=O)c2c1Sc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)c(F)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.89
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 7.3 pIC50 TTD_MultiTarget
P04818 TYMS Homo sapiens Human PF00303 7.3 IC50 ChEMBL;BindingDB
C3SWJ7 thyA Escherichia coli Pathogen PF00303 6.1 IC50 ChEMBL;BindingDB