Molecule Details
InChIKeyLTAXPWDTMINWRK-UHFFFAOYSA-N
Compound Name6-fluoro-2-(1H-imidazol-5-ylmethyl)-3,4-dihydro-1H-[1]benzothiolo[2,3-c]pyridine
Canonical SMILESFc1ccc2sc3c(c2c1)CCN(Cc1c[nH]cn1)C3
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P05093 CYP17A1 Homo sapiens Human PF00067 7.6 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.2 IC50 ChEMBL;BindingDB