Molecule Details
InChIKeyLSHYTYHPKFOCBP-UHFFFAOYSA-N
Compound Name6-(azetidin-3-ylsulfonyl)-3-[2-[(4-methoxyphenyl)methyl]-1-methylindol-4-yl]-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESCOc1ccc(Cc2cc3c(-c4ccc(S(=O)(=O)C5CNC5)c(S(N)(=O)=O)c4-c4nnn[nH]4)cccc3n2C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.45
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.9 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.4 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.1 IC50 BindingDB