Molecule Details
InChIKeyLSEOXFVSQOHSDK-HXUWFJFHSA-N
Compound NameN-[4-[6-[[2-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]acetyl]amino]-4-[(5-methyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl]sulfanylphenyl]cyclopropanecarboxamide
Canonical SMILESCc1cc(Nc2nc(Sc3ccc(NC(=O)C4CC4)cc3)nn3cc(NC(=O)CN4CCC[C@@H]4CO)cc23)n[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.0 Kd ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.8 Kd ChEMBL;BindingDB
Q9UQB9 AURKC Homo sapiens Human PF00069 7.1 Kd ChEMBL;BindingDB