Molecule Details
InChIKeyLRVSISWQSCNQKL-CALCHBBNSA-N
Canonical SMILESCOc1ccc(Nc2ncc3nc(Nc4ccccc4F)n([C@H]4CC[C@@H](O)CC4)c3n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB