Molecule Details
InChIKeyLQESNGDPCQOCKO-UHFFFAOYSA-N
Compound Name3-Imidazo[1,2-a]pyridin-3-yl-4-[6-methyl-10-(piperidine-1-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]pyrrole-2,5-dione
Canonical SMILESCc1cc2c3c(c1)c(C1=C(c4cnc5ccccn45)C(=O)NC1=O)cn3CCN(C(=O)N1CCCCC1)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P05771 PRKCB Homo sapiens Human PF00130 PF00168 PF00069 PF00433 6.4 IC50 ChEMBL;BindingDB