Molecule Details
InChIKeyLPKOEWTZGVUEJF-BQYQJAHWSA-N
Compound NameImidazo[1,2-c]pyrimidine-8-carboxamide, 27
Canonical SMILESCOc1cc(Nc2nc(NCc3ccc(/C=C/C(=O)O)cc3)n3ccnc3c2C(N)=O)cc(OC)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43403 ZAP70 Homo sapiens Human PF07714 PF00017 7.3 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 6.2 IC50 ChEMBL;BindingDB
Q15046 KARS1 Homo sapiens Human PF00152 PF01336 6.2 IC50 ChEMBL