Molecule Details
InChIKeyLPJUSCDLIIKTBR-UHFFFAOYSA-N
Compound Name6-chloro-N-[6-[(2-chloro-3-pyridinyl)oxy]-3-pyridinyl]-5-methyl-2,3-dihydroindole-1-carboxamide
Canonical SMILESCc1cc2c(cc1Cl)N(C(=O)Nc1ccc(Oc3cccnc3Cl)nc1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB