Molecule Details
InChIKeyLPIJJPHNJFECSA-UHFFFAOYSA-N
Compound Name7-(4-Fluorophenyl)-2-((3-fluoropyridin-2-yl) methyl)-8-(quinolin-6-yl)-[l,2,4]triazolo[l,5-c] pyrimidin-5-amine
Canonical SMILESNc1nc(-c2ccc(F)cc2)c(-c2ccc3ncccc3c2)c2nc(Cc3ncccc3F)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.4 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB