Molecule Details
InChIKeyLNWXGYVVZJDLCP-CYBMUJFWSA-N
Compound Name(R)-2-amino-N-(4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)phenylsulfonyl)-3-hydroxypropanamide
Canonical SMILESNc1nc(Nc2ccc(S(=O)(=O)NC(=O)[C@H](N)CO)cc2)nn1C(=O)c1c(F)cccc1F
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.85
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget