Molecule Details
InChIKeyLNNWDFRSVZFSAT-HKBQPEDESA-N
Compound Name3-[(2S)-3-[4-(cyclohexanecarbonyl)piperazin-1-yl]-2-[[3-(2,4-dimethoxyphenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide
Canonical SMILESCOc1ccc(-c2cccc(S(=O)(=O)N[C@@H](Cc3cccc(C(=N)N)c3)C(=O)N3CCN(C(=O)C4CCCCC4)CC3)c2)c(OC)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.2
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5Y6 ST14 Homo sapiens Human PF00431 PF00057 PF01390 PF00089 7.4 Ki ChEMBL;BindingDB
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.0 Ki ChEMBL;BindingDB