Molecule Details
InChIKeyLMZRJJTWTQNOEI-UHFFFAOYSA-N
Compound NameN-[4-bromo-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(5-oxopyrazolo[1,5-a]pyrimidin-4-yl)acetamide
Canonical SMILESO=C(Cn1c(=O)ccn2nccc12)Nc1scc(Br)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.78
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB