Molecule Details
InChIKeyLMNXBEZQGBWMMY-UHFFFAOYSA-N
Compound Name4-[6-[3-Chloro-4-(2-piperidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline
Canonical SMILESClc1cc(-c2cnc3c(-c4ccnc5ccccc45)cnn3c2)ccc1OCCN1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q04771 ACVR1 Homo sapiens Human PF01064 PF07714 PF08515 7.2 IC50 ChEMBL;BindingDB
P37023 ACVRL1 Homo sapiens Human PF07714 PF08515 7.0 IC50 ChEMBL;BindingDB
O00238 BMPR1B Homo sapiens Human PF01064 PF07714 PF08515 6.7 IC50 ChEMBL;BindingDB