Molecule Details
InChIKeyLMJTUYSCJIQXFP-KTPANICASA-N
Compound Name3,5-Dichloro-N-{(R)-3-(3,4-dichloro-phenyl)-2-[(Z)-methoxyimino]-5-[4-(3-methylcarbamoylmethyl-2-oxo-tetrahydro-pyrimidin-1-yl)-piperidin-1-yl]-pentyl}-N-methyl-benzamide
Canonical SMILESCNC(=O)CN1CCCN(C2CCN(CC[C@@H](/C(CN(C)C(=O)c3cc(Cl)cc(Cl)c3)=N/OC)c3ccc(Cl)c(Cl)c3)CC2)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P29371 TACR3 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB