Molecule Details
InChIKeyLMGSQMQVUYDBRD-DPUDNOKTSA-N
Compound Name(2S)-2-[[4-[(Z)-1-cyano-2-pyridin-3-ylethenyl]-2-(2-methylphenyl)benzoyl]amino]-4-methylsulfanylbutanoic acid
Canonical SMILESCSCC[C@H](NC(=O)c1ccc(/C(C#N)=C/c2cccnc2)cc1-c1ccccc1C)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.23
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.2 IC50 ChEMBL