Molecule Details
InChIKeyLMGRXYCLENIEMO-UHFFFAOYSA-N
Compound Name2-[4-[[(6,7-dimethoxy-2-methylquinolin-4-yl)amino]methyl]piperidin-1-yl]-N-hydroxypyrimidine-5-carboxamide
Canonical SMILESCOc1cc2nc(C)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 8.5 IC50 ChEMBL;BindingDB
Q96KQ7 EHMT2 Homo sapiens Human PF00023 PF12796 PF21533 PF05033 PF00856 8.1 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.6 IC50 ChEMBL;BindingDB