Molecule Details
InChIKeyLMBOMGUIBWYBDA-UHFFFAOYSA-N
Compound Name4-[1-[3-[[1-(Trifluoromethyl)cyclobutanecarbonyl]amino]cyclohexa-1,3-dien-1-yl]ethylamino]quinazoline-8-carboxamide
Canonical SMILESCC(Nc1ncnc2c(C(N)=O)cccc12)C1=CC(NC(=O)C2(C(F)(F)F)CCC2)=CCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.4 IC50 ChEMBL;BindingDB