Molecule Details
InChIKeyLKZXAQZZOSZHLE-UHFFFAOYSA-N
Compound Name3-[4-(4-methylpiperazin-1-yl)phenyl]-N-[(1-morpholin-4-ylcyclohexyl)methyl]-1H-indazole-5-carboxamide
Canonical SMILESCN1CCN(c2ccc(-c3n[nH]c4ccc(C(=O)NCC5(N6CCOCC6)CCCCC5)cc34)cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 6.4 IC50 ChEMBL
Q9NQS7 INCENP Homo sapiens Human PF03941 PF12178 6.4 IC50 ChEMBL