Molecule Details
InChIKeyLKZPAYSWYUKKEK-UHFFFAOYSA-N
Compound Name1-[6-(3-Methoxypiperidin-3-yl)-2-pyridinyl]-6-(6-methylpyrazin-2-yl)pyrazolo[4,3-c]pyridine
Canonical SMILESCOC1(c2cccc(-n3ncc4cnc(-c5cncc(C)n5)cc43)n2)CCCNC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.8 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.6 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.8 Ki ChEMBL;BindingDB