Molecule Details
InChIKeyLKXBYRYJOKCGTP-UHFFFAOYSA-N
Compound NameN-[6-cyano-1-[(3-methylimidazol-4-yl)methyl]-3,4-dihydro-2H-quinolin-3-yl]-N-methylpyridine-2-sulfonamide
Canonical SMILESCN(C1Cc2cc(C#N)ccc2N(Cc2cncn2C)C1)S(=O)(=O)c1ccccn1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.51
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.5 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.5 IC50 ChEMBL