Molecule Details
InChIKeyLKUQDQOKQYEING-UHFFFAOYSA-N
Compound NameN'-[3-methoxy-5-[3-propan-2-yl-5-[(1-propan-2-ylpiperidin-4-yl)methoxy]-1H-pyrrolo[3,2-b]pyridin-2-yl]-2-pyridinyl]methanimidamide
Canonical SMILESCOc1cc(-c2[nH]c3ccc(OCC4CCN(C(C)C)CC4)nc3c2C(C)C)c[nH]/c1=N\C=N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYK1 TLR7 Homo sapiens Human PF13855 PF01582 9.1 IC50 ChEMBL;BindingDB
Q9NR97 TLR8 Homo sapiens Human PF13855 PF01582 8.5 IC50 ChEMBL;BindingDB
Q9NR96 TLR9 Homo sapiens Human PF18837 PF13516 PF13855 PF01582 6.0 IC50 ChEMBL;BindingDB