Molecule Details
InChIKeyLKLIRPMEYRVLFV-UHFFFAOYSA-N
Compound Name3-[[4-(5-Hydroxy-2-methylanilino)pyrimidin-2-yl]amino]benzenesulfonamide
Canonical SMILESCc1ccc(O)cc1Nc1ccnc(Nc2cccc(S(N)(=O)=O)c2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P42681 TXK Homo sapiens Human PF07714 PF00017 PF00018 9.4 IC50 ChEMBL
P07948 LYN Homo sapiens Human PF07714 PF00017 PF00018 9.0 IC50 ChEMBL
P43405 SYK Homo sapiens Human PF07714 PF00017 8.4 IC50 ChEMBL