Molecule Details
InChIKeyLJUHMEDWYHTVAZ-UHFFFAOYSA-N
Compound Name3-(2''-Propylaminocarbonylsulfamoyl-biphenyl-4-ylmethyl)-5-methylsulfanyl-2-propyl-3H-imidazole-4-carboxylic acid
Canonical SMILESCCCNC(=O)NS(=O)(=O)c1ccccc1-c1ccc(Cn2c(CCC)nc(SC)c2C(=O)O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 9.5 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB