Molecule Details
InChIKeyLIUQLADXKRFWMD-UHFFFAOYSA-N
Canonical SMILESCN1CCC(COc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(C(F)(F)F)cc6)CC(C)(C)CC5)CC4)cc3Oc3cnc4[nH]ccc4c3)cc2[N+](=O)[O-])C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.45
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 9.1 IC50 ChEMBL;BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 7.8 IC50 ChEMBL;BindingDB