Molecule Details
InChIKeyLIIRZRQVACDFBI-HOTGVXAUSA-N
Compound NameN-[3-(3-Phenylisoxazol-5-Yl)propanoyl]-L-Alpha-Glutamyl-L-Alpha-Glutamyl-Amide
Canonical SMILESNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)CCc1cc(-c2ccccc2)no1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P22894 MMP8 Homo sapiens Human PF00045 PF00413 PF01471 7.0 Ki ChEMBL;BindingDB
P39900 MMP12 Homo sapiens Human PF00045 PF00413 PF01471 6.9 Ki ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 6.1 Ki ChEMBL;BindingDB