Molecule Details
InChIKeyLHMLJRCNGQZNHL-UHFFFAOYSA-N
Compound Name4-[3-(difluoromethoxy)-4-fluorophenyl]-1-(1H-pyrazol-5-ylmethyl)pyrazole
Canonical SMILESFc1ccc(-c2cnn(Cc3cc[nH]n3)c2)cc1OC(F)F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 8.1 IC50 ChEMBL;BindingDB
Q13224 GRIN2B Homo sapiens Human PF01094 PF00060 PF10613 PF10565 6.4 IC50 ChEMBL;BindingDB