Molecule Details
InChIKeyLHABRXRGDLASIH-UHFFFAOYSA-N
Compound Name5-fluoro-N-[2-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-1H-indole-2-carboxamide
Canonical SMILESO=C(NCCN1CCC(n2c(=O)[nH]c3ccccc32)CC1)c1cc2cc(F)ccc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.8
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13393 PLD1 Homo sapiens Human PF00169 PF00614 PF13091 PF00787 7.9 IC50 ChEMBL;BindingDB
O14939 PLD2 Homo sapiens Human PF00614 PF13091 PF00787 7.7 IC50 ChEMBL;BindingDB