Molecule Details
InChIKeyLGQKIASGYQMERJ-UHFFFAOYSA-N
Compound NameN-(2-(1H-imidazol-4-yl)ethyl)-6-(benzo[d][1,3]dioxol-5-yl)quinazolin-4-amine
Canonical SMILESc1nc(NCCc2c[nH]cn2)c2cc(-c3ccc4c(c3)OCO4)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HAZ1 CLK4 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB
P49759 CLK1 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB