Molecule Details
InChIKeyLGPOBVLZHCYRKV-UHFFFAOYSA-N
Compound Name4-amino-N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]-3-bromobenzenesulfonamide
Canonical SMILESCOc1cc(N)c(Cl)cc1C(=O)CCC1CCN(CCNS(=O)(=O)c2ccc(N)c(Br)c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P50406 HTR6 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB