Molecule Details
InChIKeyLGKMEHLZMDCMTK-HDYFOKATSA-N
Compound Name(10R,13S)-17-[di(propan-2-yl)carbamoyl]-10,13-dimethyl-6,7,8,9,11,12,14,15-octahydro-1H-cyclopenta[a]phenanthrene-3-carboxylic acid
Canonical SMILESCC(C)N(C(=O)C1=CCC2C3CCC4=CC(C(=O)O)=CC[C@]4(C)C3CC[C@]12C)C(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.15
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.2 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 8.2 pIC50 TTD_MultiTarget