Molecule Details
InChIKeyLFQCICBMIDNCDI-UHFFFAOYSA-N
Compound Name2-(Dimethylamino)-1-[4-[6-[[5-fluoro-4-(8-fluoro-4-propan-2-yl-2,3-dihydro-1,4-benzoxazin-6-yl)pyrimidin-2-yl]amino]-3-pyridinyl]piperidin-1-yl]ethanone
Canonical SMILESCC(C)N1CCOc2c(F)cc(-c3nc(Nc4ccc(C5CCN(C(=O)CN(C)C)CC5)cn4)ncc3F)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00534 CDK6 Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 6.7 IC50 ChEMBL;BindingDB