Molecule Details
InChIKeyLFAGGDAZZKUVKO-JAGWWQSPSA-N
Compound Name(1R,2R,3R,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Canonical SMILESN[C@]1(C(=O)O)[C@H]2[C@@H](C[C@H]1OCc1ccc(Cl)c(Cl)c1)[C@]2(F)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q14416 GRM2 Homo sapiens Human PF00003 PF01094 PF07562 8.2 IC50 ChEMBL;BindingDB
Q14832 GRM3 Homo sapiens Human PF00003 PF01094 PF07562 8.0 IC50 ChEMBL;BindingDB