Molecule Details
InChIKeyLEZLIAHSOVEHCJ-HXUWFJFHSA-N
Compound NamePyrimidylpyrrole, 9f
Canonical SMILESCc1cnc(Nc2ccccc2O)nc1-c1c[nH]c(C(=O)N[C@H](CO)c2ccccc2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 8.4 Ki ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 7.0 Ki ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget