Molecule Details
InChIKeyLEMPHOJARYISJD-UHFFFAOYSA-N
Compound Name3-methylbutyl N-[2-[3-fluoro-4-[[2-methyl-4-oxo-6-(propan-2-ylcarbamoylamino)quinazolin-3-yl]methyl]phenyl]phenyl]sulfonylcarbamate
Canonical SMILESCc1nc2ccc(NC(=O)NC(C)C)cc2c(=O)n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)OCCC(C)C)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P50052 AGTR2 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P30556 AGTR1 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB