Molecule Details
InChIKeyLDXWEXQSCRPNPG-UHFFFAOYSA-N
Compound Name5-(4-Chlorophenyl)-n-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propyl)-2-methyl-1h-pyrrole-3-carboxamide hydrochloride
Canonical SMILESCc1[nH]c(-c2ccc(Cl)cc2)cc1C(=O)NCCCN1CCN(c2cccc(Cl)c2Cl)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.2 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB