Molecule Details
InChIKeyLDWBULFGVRAVMR-UHFFFAOYSA-N
Compound Name2-N-[(4-chloro-1H-benzimidazol-5-yl)methyl]-4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-2-N-methylpyrimidine-2,4-diamine
Canonical SMILESCN(Cc1ccc2[nH]cnc2c1Cl)c1nccc(Nc2cc(C3CC3)[nH]n2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.5 Ki ChEMBL;BindingDB
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 8.3 Ki ChEMBL;BindingDB
O96013 PAK4 Homo sapiens Human PF00786 PF00069 6.6 Ki ChEMBL;BindingDB