Molecule Details
InChIKeyLCYPGGDZOSRDEW-LHSJRXKWSA-N
Compound Name(3R)-N-[(3S)-1-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperidin-3-yl]-2,3-dihydro-1,4-benzodioxine-3-carboxamide
Canonical SMILESCOc1cc2nc(N3CCC[C@H](NC(=O)[C@H]4COc5ccccc5O4)C3)nc(N)c2cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB