Molecule Details
InChIKeyLCTLPROJUJRGOK-OYGGHGNESA-N
Compound Name3-(5-(hexa-2,4-dienylidene)-2-oxo-5,6-dihydro-2H-pyran-3-yl)-N-hydroxypropanamide
Canonical SMILESC/C=C/C=C\C=C1\C=C(CCC(=O)NO)C(=O)OC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.2 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 7.6 IC50 ChEMBL;BindingDB
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 7.5 IC50 ChEMBL;BindingDB